中华医学超声杂志

应用化学 ›› 1990, Vol. 0 ›› Issue (6): 54-57.

• 研究简报 • 上一篇    下一篇

一些嘧啶酰胺的合成及其生物活性

于中生, 陈馥衡   

  1. 北京农业大学应用化学研究所 北京 100094
  • 收稿日期:1989-11-15 修回日期:1990-05-10 出版日期:1990-12-10 发布日期:1990-12-10

SYNTHESIS OF AMIDE CONTAINING PYRIMIDINES AND THEIR BIOACTIVITY

Yu Zhongsheng, Chen Fuheng   

  1. Institute of Applied Chemistry, Beijing Agricultural University, Beijing 100094
  • Received:1989-11-15 Revised:1990-05-10 Published:1990-12-10 Online:1990-12-10

PDF

338

被引次数

9 | 1

摘要： 嘧啶环是生物活性化合物中具有较好生理活性的基因[1]。本文试图将嘧啶环引入农用药剂,合成系列酰胺类化合物。生物试验结果表明,其中一些化合物具有杀蝇效能,一些化合物对较难防治的寄生疫霉具有良好的抑制效能。

关键词: 嘧啶, 酰胺, 杀虫作用, 杀菌活性, 合成

Abstract: Amide derivatives[containing pyrimidine group have been synthesized with generalformula where R1 = H, CH3; R1 = CH3, C6H5, CH3C6H5, CH3OC6H4, ClC6H4, FC6H4 The structures of the compounds were confirmed by IR, 1H-NMR and elemental analy-sis. Some of the compounds are effective against Musca domestica and fungi.

Key words: pyrimidine amide, insecticidal activity, fungicidal activity, synthesis

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