[1] | Pirhadi S,Shiri F,Ghasemi J B. Methods and Applications of Structure-based Pharmacophores in Drug Discovery[J]. Curr Top Med Chem,2013,13(9):1036-1047. | [2] | GUO Zongru. Strategy of Molecular Drug Design: Activity and Druggability[J]. Acta Pharm Sin,2010,45(5):539-547(in Chinese). 郭宗儒. 药物分子设计与策略:药理活性与成药性[J]. 药学学报,2010,45(5):539-547. | [3] | Suresh N,Nagesh HN,Sekhar KV,et al.Synthesis of Novel Ciprofloxacin Analogues and Evaluation of Their Anti-proliferative Effect on Human Cancer Cell Lines[J]. Bioorg Med Chem Lett,2013,23(23):6292-6295. | [4] | WANG Guoqiang,DUAN Nannan,CAO Tieyao,et al.Antitumor Fluoroquinolone C3-Isostere Derivatives(Ⅰ)—Synthesis and Activity of Bis-oxadiazole Methyl-sulfide Derivatives[J]. Chinese J Appl Chem,2012,29(7):769-774(in Chinese). 王国强,段楠楠,曹铁耀,等. 抗肿瘤氟喹诺酮 C3等排衍生物(Ⅰ)—双噁二唑甲硫醚衍生物的合成和抗肿瘤活性[J]. 应用化学,2012,29(7):769-774. | [5] | XIE Songqiang,CHEN Yinsheng,WANG Guoqiang,et al.Part Ⅳ.Synthesis and Antitumor Evaluation of s-Triazolothiadiazines and Pyrazolo s-Triazoles Derived From Ciproxacin[J]. Acta Pharm Sin,2012,47(1):66-71(in Chinese). 谢松强,陈寅生,王国强,等. Part Ⅳ. 环丙沙星C-3羧基衍生物均三唑并噻二嗪及吡唑并均三唑的合成和抗肿瘤活性研究[J]. 药学学报,2012,47(1):66-71. | [6] | Megally Abdo N Y,Kamel M M. Synthesis and Anticancer Evaluation of 1,3,4-Oxadiazoles, 1,3,4-Thiadiazoles, 1,2,4-Triazoles and Mannich Bases[J]. Chem Pharm Bull(Tokyo),2015,63(5):369-376. | [7] | Huang H,Chen Q,Ku X,et al.A Series of Alpha-heterocyclic Carboxaldehyde Thiosemicarbazones Inhibit Topoisomerase II Alpha Catalytic Activity[J]. J Med Chem,2010,53(8):3048-3064. | [8] | XU Qiuju,Hou Lili,WU Zhaofeng,et al.Synthesis and Antitumor Evaluation of Fluoroquinolon C3 s-Triazole Oxadiazole Methylsulfide Derivatives of Ofloxacin[J]. Chinese Pharm J,2014,49(7):609-612(in Chinese). 许秋菊,侯莉莉,仵钊锋,等. 氟喹诺酮C3 均三唑噁二唑甲硫醚衍生物的合成及抗肿瘤活性[J]. 中国药学杂志,2014,49(7):609-612. |
|